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Principals, terminologystationery phase,mobile phase, classificationofchromatographymethods,migrationrateofspecies (partitioncoefficient,retentiontime,adjustedretentiontime),Rateofsolutemigration(capacityfactor,selectivityfactor),Columnefficiencyandbandbroadening(shapeof peakGausssian, plate height, number of theoretical plates, vanDeemeter equation), Optimisation of column performance (Columnresolution, capacity factor, selective factor, tailing factor, peak width),Qualitative analysis, Quantitative analysis (Peak height, peak areas,calibrationandinternalstandard,externalstandard,areanormalization).Ģ. TheOrganicChemistryofDrugSynthesis,DanielLednicer,Vols1to7,Wiley. PharmaceuticalChemistry.J.Roth,A.KleemanandT.Beissewenger,EllisHorwoodLtd.1988.Ħ.
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Johnson and Jie Jack Li, WileyInterscience,2007.ĥ. Medicinal Chemistry, Ashutosh Kar, 4th Edition, New Age International Publishers,2007.Ĥ. Williams.Williams&Wilkins,Baltimore,2002.ģ. Foyes Principals of Medicinal Chemistry, Eds. WilsonandGisvoldsTextbookofOrganicMedicinalandPharmaceuticalChemistry.Beale,LippincottWilliams&Wilkins,2004Ģ. (iv) VasodilatorsandKchannelagonists(diazoxide,minoxidil)(v) Antihyperlipidemic agents (clofibrate*, gemfibrozil, niacin, lovastatin,Ītorvastatin) 3*Indicatessynthesistobediscussedġ. (iii)Antihypertensiveagents(a)reviewofadrenergicagents(b)reviewofCa channel blockers (c) ACE inhibitors (captopril*, enalapril,benzepril, ramipril) (d) angiotensin II receptor antagonists (losartan,valsartan*,candersartan) (ii) antiarrhythmic agents (quinidine, procainamide*, disopyramide,lidocaine, tocainide,mexilitine, encainide, amiodarone, pro[afenone,verapamil,diltiazen,propranolol,sotalol*). Tetranitrate, verapamil, bepridil, diltiazem, nifendipine*, amlodipine,nimodipine,dipyridamole) CVSDrugs:(i) antianginal agents (amyl nitrite, isosorbide dinitrate, pentaerythritol Phenoxybenzamine,prazosin,doxazosin)(iv) adrenergic antagonists (propranolol*, atenolol, metoprolol,Īcebutalol,alprenolol,timolol,labetalol*)other adrenergic agents (amphetamine, pseudophedrine,ephedrine,guanethidine*,propylhexedrine,reserpine).ģ. Isoxsuprine,ritodrine)(iii)adrenergic antagonists (tolazine, phentolamine, Oxymetazoline,methyldopa,clonidine*,guanabenz,guanfacine)(ii) adrenergicagonists(isoproternol,terbutaline*,albuterol,salmeterol, AdrenergicDrugs:(i) adrenergic agonists (phenylephrine, naphazoline, xylometazoline,
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(iv)Ganglionblockingagents(trimethaphan,camsylate,mecamylamine)(v) Neuromuscularblockingagents(tubocurarine,gallamine,triethiodide,Ģ. Hydrobromide, ipratropium bromide) synthetic cholinergicantagonists (cyclopentolate*, dicyclomine*, ben/otropine mesylate,procyclidinehydrochloride,isopropamideiodide,tropicamide) Pilocarpine)(ii) Ach esterase inhibitors (physostigmine, neostigmine*,tacrine*,Īmbenoniumchloride,isofluorphate,pralidoxime)(iii)Cholinergic antagonists (atropine, scopolamine, homatropine CholinergicDrugs:(i) cholinergic agonists (methocholine, carbochol*, bethanechol, Topic HoursDiscussion of the following classes of drugs including classification,chemical nomenclature, structure including stereochemistry, genericnames, chemistry, physicochemical properties, SAR, metabolism,molecular mechanism of action and synthesis, introduction to rationaldevelopmentifanyoftheclassofdrugs.ġ. PHARMACEUTICALMEDICINALCHEMISTRYIII 3hrs/week SYLLABUSCOPYFORFINALYEARB.PHARMSEMSETERVII